KR-32568
目录号 : KCM15444
CAS No. : 852146-73-7
纯度 : ≥98%
KR-32568 is an inhibitor of the sodium-hydrogen exchanger isoform-1 (NHE-1; IC = 230 nM). It restores cardiac contractile function ex vivo in an isolated ischemic rat heart model when used at a concentration of 10 μM. KR-32568 (0.3 mg/kg) reduces myocardial infarct size in a rat model of ischemia and reperfusion injury.
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分子式 |
C13H12FN3O2
|
分子量 |
261.3
|
CAS号 |
852146-73-7
|
中文名称 |
N-(diaminomethylidene)-5-(5-fluoro-2-methylphenyl)furan-2-carboxamide
|
储存方式 |
-20°C
|