M40 是一个有效的，非竞争性的 galanin receptor 拮抗剂。
| 生物活性 |
M40 is a potent, non-selective galanin receptor antagonist. |
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| 体外研究 |
M40 (1 μM) displaces [mono[IJodo-Tyr]galanin from binding sites in the hippocampus, hypothalamus, and spinal cord. M40 has a lower affinity than galanin for all membranes. The IC50 values are 6 nM in the hippocampus, 15 nM in the hypothalamus, 12 nM in the spinal cord, and 3 nM in the insulinoma cells. M40 (1 μM) completely blocks I-labeled galanin-binding sites. |
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| 分子式 |
C94H145N23O24
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| 分子量 |
1980.31
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| CAS号 |
143896-17-7
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
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客服小K 
客服小K
Data Sheet
